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Letters in Drug Design & Discovery

ISSN (Print): 1570-1808
ISSN (Online): 1875-628X

Latest Issue: Volume 17 , Issue 11 , 2020

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Volume 17, Issue 11


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Page: 1329-1329
Author: György Keglevich
Doi: 10.2174/157018081711201002154128

Research Article

Design, Synthesis, Docking and Computational Pharmacokinetic Profiling of New Pyrazolinyl Thiazolinone Biheterocycles as Potent Antimicrobial Agents

Page: 1342-1354
Author: Vinutha Vittala Salian, Badiadka Narayana*, Balladka Kunhanna Sarojini, Sharath Chandra Kodandoor and Anupam Glorious Lobo
Doi: 10.2174/1570180817999200623115049

Research Article

Evaluating Phenyl Propanoids Isolated from Citrus Medica as Potential Inhibitors for Mitotic kinesin Eg5

Page: 1355-1363
Author: Himesh Makala, Venkatasubramanian Ulaganathan*, Aravind Sivasubramanian, Narendran Rajendran and Shankar Subramanian
Doi: 10.2174/1570180817999200630125449

Research Article

QSAR Studies of Sulfonamide Hydroxamates Derivatives as MMP-2 Inhibitors Topomer CoMFA and Molecular Docking

Page: 1364-1371
Author: Jian-Bo Tong*, Feng Yi, Ding Luo and Tian-Hao Wang
Doi: 10.2174/1570180817999200630124920

Research Article

Synthesis, Characterization and Antimicrobial Activity of Some Novel 1- substituted Benzimidazole Derivatives

Page: 1372-1379
Author: Erkut Isik, Demet Astley, Seda Yuksekdanaci* and Ihsan Yasa
Doi: 10.2174/1570180817999200531164230

Research Article

Design, Synthesis, In vitro and In silico Evaluation of New Hydrazonebased Antitumor Agents as Potent Akt Inhibitors

Page: 1380-1392
Author: Emine Merve Güngör, Mehlika Dilek Altıntop*, Belgin Sever and Gülşen Akalın Çiftçi
Doi: 10.2174/1570180817999200618163507

Research Article

Evaluation of Kaempferol as AKT Dependent mTOR Regulator via Targeting FKBP-12 in Hepatocellular Carcinoma: an In silico Approach

Page: 1401-1408
Author: Pooja Siniprasad, Bhagyalakshmi Nair, Vaisali Balasubramaniam, Prashanth Sadanandan, Puliyapally Krishnan Namboori and Lekshmi Reghu Nath*
Doi: 10.2174/1570180817999200623115703

Research Article

Synthesis and Evaluation of Dapagliflozin Ester Prodrugs with Improved Hygroscopicity and Thermal Stability

Page: 1409-1421
Author: Si Young Sung, Yu Na Chae, Dae Young Lee, Kyeong Min Kim, Eun Jung Kim, Ji Hye Han, Wook Kim and Sung-Hwa Yoon*
Doi: 10.2174/1570180817999200618162949

Research Article

Comparative Proteome Analysis of Mycobacterium Tuberculosis Strains - H37Ra, H37Rv, CCDC5180, and CAS/NITR204: A Step Forward to Identify Novel Drug Targets

Page: 1422-1431
Author: Shradheya R.R. Gupta, Ekta Gupta, Avnam Ohri, Sandeep Kumar Shrivastava, Sumita Kachhwaha, Vinay Sharma, Rupesh Kumar Mishra and Ravi Ranjan Kumar Niraj*
Doi: 10.2174/1570180817999200531165148

Research Article

Novel 2-(5-Aryl)thiophen-2-yl)benzimidazoles; Design, Synthesis and In vitro Evaluation Against Cercarial Phase of Schistosoma mansoni

Page: 1432-1438
Author: Serry Atta El Bialy, Basem Mansour*, Waleed Abdelhakeem Bayoumi, Amira Taman and Hassan Mohammed Eissa
Doi: 10.2174/1570180817999200523181211

Research Article

High Anti-cancer Activity, Low Animal Toxicity, and Structure Activity Relationships of Curcumin Analogs

Page: 1439-1455
Author: Sen-Chuan Song, Yu-Liang Mai, Hua-Hong Shi, Bing Liao* and Fei Wang*
Doi: 10.2174/2352096513999200714103641

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